Molecule Details
InChIKeyQFRIGJQJVRCBFQ-HNNXBMFYSA-N
Compound NameN-[4-bromo-3-[(3R)-3-cyclopropylpyrrolidin-1-yl]sulfonylphenyl]-2-(5-methyl-6,7-dihydro-4H-triazolo[4,5-c]pyridin-1-yl)acetamide
Canonical SMILESCN1CCc2c(nnn2CC(=O)Nc2ccc(Br)c(S(=O)(=O)N3CC[C@H](C4CC4)C3)c2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BXF3 CECR2 Homo sapiens Human PF00439 8.0 IC50 ChEMBL;BindingDB
Q92830 KAT2A Homo sapiens Human PF00583 PF00439 PF06466 6.8 Kd ChEMBL;BindingDB
P21675 TAF1 Homo sapiens Human PF00439 PF12157 PF09247 PF15288 6.7 IC50 ChEMBL;BindingDB