Molecule Details
InChIKeyQFPXEFZKXYSMPH-UHFFFAOYSA-N
Compound Name5-Methyl-1-[2-(pyridin-2-ylmethyloxy)3-methylpyridin-5-ylcarbamoyl]-6-trifluoromethylindoline
Canonical SMILESCc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1cnc(OCc3ccccn3)c(C)c1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB