Molecule Details
InChIKeyQFPUYOAZKKYGQE-CHWSQXEVSA-N
Compound Name5-fluoro-4-((R)-1-(3-fluorophenyl)propan-2-yloxy)-2-((R)-2-methylpiperazin-1-yl)pyrimidine
Canonical SMILESC[C@H](Cc1cccc(F)c1)Oc1nc(N2CCNC[C@H]2C)ncc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P05177 CYP1A2 Homo sapiens Human PF00067 6.4 IC50 ChEMBL;BindingDB