Molecule Details
InChIKeyQFMZANLICXRGCX-RFAUZJTJSA-N
Compound Name4''-[(4R,5S)-4-methyl-2-oxo-1,3-oxazolidin-5-yl]-2-(1H-tetrazol-5-yl)biphenyl-3-sulfonamide
Canonical SMILESC[C@H]1NC(=O)O[C@H]1c1ccc(-c2cccc(S(N)(=O)=O)c2-c2nnn[nH]2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.52
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.2 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.4 IC50 BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 8.0 IC50 BindingDB