Molecule Details
InChIKeyQFGVLITXAHSQBT-UHFFFAOYSA-N
Compound Name5-(4-Acetyl-1,4-diazepan-1-yl)-5-(4-phenoxyphenyl)-1,3-diazinane-2,4,6-trione
Canonical SMILESCC(=O)N1CCCN(C2(c3ccc(Oc4ccccc4)cc3)C(=O)NC(=O)NC2=O)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.68
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.8 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.5 pIC50 TTD_MultiTarget