Molecule Details
InChIKeyQERDWLFJAPHTPD-DPODCYPTSA-N
Compound NameN-benzyl-N-(((4R,4aS,6R,7R,7aR,12bS)-3-(cyclopropylmethyl)-7,9-dimethoxy-1,2,3,4,5,6,7,7a-octahydro-4a,7-ethano-4,12-methanobenzofuro[3,2-e]isoquinolin-6-yl)methyl)acetamide
Canonical SMILESCOc1ccc2c3c1O[C@H]1[C@@]4(OC)CC[C@@]5(C[C@@H]4CN(Cc4ccccc4)C(C)=O)[C@@H](C2)N(CC2CC2)CC[C@]315
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.8 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB