Molecule Details
InChIKeyQEJJXMNBAFWGJK-UHFFFAOYSA-N
Compound Name2-[[3-[(4-fluorophenyl)methoxy]azetidin-1-yl]methyl]-7-(oxan-4-yl)-3H-imidazo[5,1-f][1,2,4]triazin-4-one
Canonical SMILESO=c1[nH]c(CN2CC(OCc3ccc(F)cc3)C2)nn2c(C3CCOCC3)ncc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O76083 PDE9A Homo sapiens Human PF00233 8.0 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 6.0 IC50 ChEMBL
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 6.0 IC50 ChEMBL