Molecule Details
InChIKeyQEILUNIAOIINON-QFIPXVFZSA-N
Compound Name(2S)-2-amino-3-(1H-indol-3-yl)-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]propanamide
Canonical SMILESN[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCCNc1c2c(nc3ccccc13)CCCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.4 IC50 ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 6.2 IC50 ChEMBL;BindingDB