Molecule Details
InChIKeyQEEMJZXDEIFDDR-ZRUFSTJUSA-N
Compound Name(2S)-2-[[(2S,5R)-2-[[(2S)-4,4-difluoropyrrolidin-2-yl]methoxycarbamoyl]-3-methyl-7-oxo-1,6-diazabicyclo[3.2.1]oct-3-en-6-yl]oxy]-2-fluoroacetic acid
Canonical SMILESCC1=C[C@@H]2CN(C(=O)N2O[C@@H](F)C(=O)O)[C@@H]1C(=O)NOC[C@@H]1CC(F)(F)CN1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.0
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00811 ampC Escherichia coli (strain K12) Pathogen PF00144 7.4 IC50 ChEMBL;BindingDB
P62593 bla Escherichia coli Pathogen PF13354 7.0 IC50 BindingDB
Q6XEC0 OXA-48 Klebsiella pneumoniae Pathogen PF00905 6.6 IC50 BindingDB