Molecule Details
InChIKeyQEBCPSVFPDGMJX-UHFFFAOYSA-N
Compound Name2-[[4-[2-(2-methylquinolin-5-yl)oxyethyl]piperazin-1-yl]methyl]-7H-1,2-benzoxazin-6-one
Canonical SMILESCc1ccc2c(OCCN3CCN(CN4C=CC5=CC(=O)CC=C5O4)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB