Molecule Details
InChIKeyQCQCMNUQTMIKHU-UHFFFAOYSA-N
Compound Name5-methyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)pyrazine-2-carboxamide
Canonical SMILESCc1cnc(C(=O)Nc2cc(-c3ccnc(Nc4ccccc4)c3)ccn2)cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB