Molecule Details
InChIKeyQCKWETFAVPLIJH-UHFFFAOYSA-N
Compound Name5-[3-(4-cyclopropylpyrimidin-2-yl)-1H-indol-5-yl]-N-(oxetan-3-yl)-1,3,4-oxadiazol-2-amine
Canonical SMILESc1cc(C2CC2)nc(-c2c[nH]c3ccc(-c4nnc(NC5COC5)o4)cc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.9 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB