Molecule Details
InChIKeyQBOWGZQRUNUQGL-ZDLGFXPLSA-N
Compound Name5-(2-fluorophenyl)-4-oxo-N-[(3Z)-2-oxo-3-(1H-pyrrol-2-ylmethylidene)-1H-indol-6-yl]-1H-pyridine-3-carboxamide
Canonical SMILESO=C1Nc2cc(NC(=O)c3c[nH]cc(-c4ccccc4F)c3=O)ccc2/C1=C/c1ccc[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 7.4 IC50 ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 7.0 IC50 ChEMBL;BindingDB