Molecule Details
InChIKeyQBMHBUSZNODSPS-UHFFFAOYSA-N
Compound Name1-(6-(6-(5-ethylpyridin-3-yl)-1H-pyrazolo[4,3-c]pyridin-1-yl)pyridin-2-yl)-1,4-diazepan-6-ol
Canonical SMILESCCc1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC(O)C3)n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.0 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.8 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB