Molecule Details
InChIKeyQBHUGPKPNMGAOH-IBGZPJMESA-N
Compound Name(3S)-N-[4-(difluoromethoxy)phenyl]-3-ethyl-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide
Canonical SMILESCC[C@]1(C)NC(=O)c2cc(S(=O)(=O)Nc3ccc(OC(F)F)cc3)ccc2NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q10469 MGAT2 Homo sapiens Human PF05060 7.6 IC50 ChEMBL;BindingDB
P26572 MGAT1 Homo sapiens Human PF03071 7.2 IC50 ChEMBL;BindingDB
Q09327 MGAT3 Homo sapiens Human PF04724 6.9 IC50 ChEMBL;BindingDB