Molecule Details
InChIKeyPZIMFNJQILPVJP-UHFFFAOYSA-N
Compound NameN-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(dimethylamino)pyridin-2-yl]pyrimidin-4-yl]acetamide
Canonical SMILESCC(=O)Nc1cc(-c2cccc(N(C)C)n2)nc(-n2nc(C)cc2C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB