Molecule Details
InChIKeyPYXVPLGVUNHGEJ-VKAKAFFBSA-N
Compound Name(3R,3aS)-7,8-Dimethoxy-3-{4-[3-(2-methoxy-phenyl)-2-methyl-allyl]-piperazin-1-ylmethyl}-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole
Canonical SMILESCOc1ccccc1/C=C(\C)CN1CCN(C[C@@H]2ON=C3c4cc(OC)c(OC)cc4OC[C@H]32)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.8 Ki ChEMBL;BindingDB