Molecule Details
InChIKeyPYWUADTVINPSEC-YVLHZVERSA-M
Compound NameSodium; 5,5,8-trioxo-3-(2-phenoxy-acetoxymethyl)-7-[1-pyridin-2-yl-meth-(Z)-ylidene]-5lambda*6*-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate
Canonical SMILESO=C(COc1ccccc1)OCC1=C(C(=O)[O-])N2C(=O)/C(=C/c3ccccn3)C2S(=O)(=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q59401 Enterobacter cloacae Pathogen PF00144 6.9 IC50 ChEMBL;BindingDB
Q6W9J1 blaTEM-1 Enterobacter cloacae Pathogen PF13354 6.1 IC50 ChEMBL
Q7B899 bla Klebsiella pneumoniae Pathogen PF13354 6.1 IC50 BindingDB