Molecule Details
InChIKeyPYUVRCPASPJQHH-UHFFFAOYSA-N
Compound Name6-Chloro-17-methyl-2-oxido-9,15-dioxo-2,14,16,17-tetraazatetracyclo[8.7.0.0;{3,8}.0;{11,16}]heptadeca-1,3,5,7,10-pentaen-2-ium
Canonical SMILESCn1c2[n+]([O-])c3ccc(Cl)cc3c(=O)c-2c2n1C(=O)NCC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.23
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.1 IC50 ChEMBL
P53779 MAPK10 Homo sapiens Human PF00069 6.1 IC50 ChEMBL