Molecule Details
InChIKeyPXYNXQORCWJBOI-UHFFFAOYSA-N
Compound Name3-[4-[4-(4-Amino-6,7-dimethoxyquinazolin-2-yl)piperazine-1-carbonyl]triazol-1-yl]-7-(diethylamino)chromen-2-one
Canonical SMILESCCN(CC)c1ccc2cc(-n3cc(C(=O)N4CCN(c5nc(N)c6cc(OC)c(OC)cc6n5)CC4)nn3)c(=O)oc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35368 ADRA1B Homo sapiens Human PF00001 9.5 IC50 ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 9.4 IC50 ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB