Molecule Details
InChIKeyPXWTVOJRXKUHBC-UHFFFAOYSA-N
Compound NameUS8835436, Example 90
Canonical SMILESCCc1c(C(=O)NCCCN2CCN(c3cccc(C)c3C)CC2)nc(-c2ccc(Cl)cc2Cl)n1-c1ccc(Br)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.5 IC50 ChEMBL;BindingDB