Molecule Details
InChIKeyPXWNTBGUQKWMOQ-UHFFFAOYSA-N
Compound Name4-Amino-6,7-dimethoxy-2-[4-(2-benzoylacetyl)-1-piperazinyl]-quinazoline
Canonical SMILESCOc1cc2nc(N3CCN(C(=O)CC(=O)c4ccccc4)CC3)nc(N)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35368 ADRA1B Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB