Molecule Details
InChIKeyPXTOBFKTYOPTQD-UHFFFAOYSA-N
Compound Name2-Amino-6-methyl-5-(2-naphthylsulfanyl)thieno[2,3-d]pyrimidin-4(3H)-one
Canonical SMILESCc1sc2nc(N)[nH]c(=O)c2c1Sc1ccc2ccccc2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.07
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.9 pIC50 TTD_MultiTarget
P04818 TYMS Homo sapiens Human PF00303 6.9 IC50 ChEMBL;BindingDB
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.4 IC50 ChEMBL;BindingDB