Molecule Details
InChIKeyPXDBZSCGSQSKST-UHFFFAOYSA-N
Compound NameEtonitazene
Canonical SMILESCCOc1ccc(Cc2nc3cc([N+](=O)[O-])ccc3n2CCN(CC)CC)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.79
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB01462
Drug NameEtonitazene
CAS Number911-65-9
Groups experimental illicit
ATC Codes nan
Descriptionnan

Categories: Heterocyclic Compounds, Fused-Ring
Cross-references: BindingDB: 50013847 CHEMBL312040 ChemSpider: 12908 Guide to Pharmacology: 1624 IUPHAR: 1624 PubChem:13493 PubChem:46508885 Wikipedia: Etonitazene ZINC: ZINC000004215955
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.9 Ki BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 6.7 Ki BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P35372 OPRM1 Mu-type opioid receptor inhibitor targets
P41143 OPRD1 Delta-type opioid receptor inhibitor targets
P41145 OPRK1 Kappa-type opioid receptor inhibitor targets