Molecule Details
InChIKeyPWVZGBVCDDZZNQ-QHCPKHFHSA-N
Compound Name(20S)-20-benzyl-8,25-dichloro-18-methyl-12-oxa-1,4,18,21,23-pentazatricyclo[20.3.1.06,11]hexacosa-6(11),7,9,22,24-pentaene-3,26-dione
Canonical SMILESCN1CCCCCOc2ccc(Cl)cc2CNC(=O)Cn2c(Cl)cnc(c2=O)N[C@@H](Cc2ccccc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 10.7 Ki ChEMBL;BindingDB
P00750 PLAT Homo sapiens Human PF00008 PF00039 PF00051 PF00089 8.5 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.4 Ki ChEMBL;BindingDB