Molecule Details
InChIKeyPWBGPHVFGDQYNG-UHFFFAOYSA-N
Compound NameN-((1H-imidazol-2-yl)methyl)-6-(benzo[d][1,3]dioxol-5-yl)quinazolin-4-amine
Canonical SMILESc1c[nH]c(CNc2ncnc3ccc(-c4ccc5c(c4)OCO5)cc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HAZ1 CLK4 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB