Molecule Details
InChIKeyPVFNDFZQGWYILU-UHFFFAOYSA-N
Compound NameN-[4-[3-(4-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]acetamide
Canonical SMILESCC(=O)Nc1ccc(-c2cnc3[nH]cc(-c4ccc(O)cc4)c3c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB