Molecule Details
InChIKeyPUWJQTDZRWOSDD-VIFPVBQESA-N
Compound Name1-N-[(2S)-3-amino-2-hydroxypropyl]-4-(2-amino-4-pyridinyl)-3-(2H-tetrazol-5-yl)benzene-1,2-disulfonamide
Canonical SMILESNC[C@H](O)CNS(=O)(=O)c1ccc(-c2ccnc(N)c2)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.31
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q2QC95 blaoxa-10 Klebsiella pneumoniae Pathogen PF00905 9.6 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.4 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.9 IC50 BindingDB