Molecule Details
InChIKeyPUMGLRKCTPGWSJ-UHFFFAOYSA-N
Compound Name2-[2-[[4-(1-Cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]amino]ethyl]guanidine
Canonical SMILESN=C(N)NCCNc1nc2ccccc2n(C2CCN(C3CCCCCCC3)CC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 8.2 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB