Molecule Details
InChIKeyPUHKAOLWMGXVFS-UHFFFAOYSA-N
Compound NameN-[5-fluoro-4-(8-fluoro-4-propan-2-yl-2,3-dihydro-1,4-benzoxazin-6-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinolin-5-amine
Canonical SMILESCC(C)N1CCOc2c(F)cc(-c3nc(Nc4cccc5c4CCNC5)ncc3F)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 7.7 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB