Molecule Details
InChIKeyPUGXENIKUPHCAF-CYBMUJFWSA-N
Compound Name4-[2-methyl-3-[(2~{R})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine
Canonical SMILESCc1nc2ccc(-c3cc(N)nc(N)c3)nc2n1C[C@@H](C)Oc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB