Molecule Details
InChIKeyPUECNZWNMCIENI-UHFFFAOYSA-N
Canonical SMILESCOc1ccc2nc(NCC(F)(F)F)c(Cc3c(=O)[nH]c(C(C)C)c4cc(OC)c(OC)cc34)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 7.3 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 6.5 IC50 ChEMBL;BindingDB