Molecule Details
InChIKeyPTTHTNNSSNKMSD-UHFFFAOYSA-N
Compound Name[5-(3-{5-[(4-fluoropiperidin-1-yl)methyl]-1H-indol-2-yl}-1H-indazol-6-yl)-1H-1,2,3-triazol-4-yl]methanamine
Canonical SMILESNCc1nn[nH]c1-c1ccc2c(-c3cc4cc(CN5CCC(F)CC5)ccc4[nH]3)n[nH]c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.67
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 10.0 IC50 ChEMBL;BindingDB
P50613 CDK7 Homo sapiens Human PF00069 6.5 IC50 ChEMBL
P51946 CCNH Homo sapiens Human PF16899 PF00134 6.5 IC50 BindingDB