Molecule Details
InChIKeyPTMZDVIBDZFFRW-JCMHNJIXSA-N
Compound Name(E)-ethyl 3-(1-(hydroxyimino)-2,3-dihydro-1H-inden-5-ylamino)thieno[2,3-c]pyridine-2-carboxylate
Canonical SMILESCCOC(=O)c1sc2cnccc2c1Nc1ccc2c(c1)CC/C2=N/O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL6.99
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 7.5 IC50 ChEMBL
P08684 CYP3A4 Homo sapiens Human PF00067 7.3 IC50 ChEMBL
P33261 CYP2C19 Homo sapiens Human PF00067 6.9 IC50 ChEMBL
P05177 CYP1A2 Homo sapiens Human PF00067 6.2 IC50 ChEMBL