Molecule Details
InChIKeyPSVLBKXIZLIMQR-UHFFFAOYSA-N
Compound Name1-(16-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Canonical SMILESCN(C)CC1CC2c3ccccc3Cc3cc(F)ccc3N2O1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 8.9 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 8.3 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB