Molecule Details
InChIKeyPSSRRSJCOUNDGG-UHFFFAOYSA-N
Compound Name4-[4-[2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Canonical SMILESO=S(=O)(c1cncc2ccccc12)N1CCC(CCN2CCN(c3cccc(F)c3)CC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL6.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P34969 HTR7 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.0 Ki ChEMBL