Molecule Details
InChIKeyPSJHTNRKPOXZIN-JTQLQIEISA-N
Compound Name8-(methyloxy)-2-[(2S)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-one
Canonical SMILESCOc1ccc2oc3c(=O)[nH]c([C@@H]4CCCN4)nc3c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P67870 CSNK2B Homo sapiens Human PF01214 6.6 IC50 ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 6.6 IC50 ChEMBL