Molecule Details
InChIKeyPSFMCOGQKUBLKM-UHFFFAOYSA-N
Compound Name8-Methyl-2-methylsulfanyl-9-propan-2-ylpyrrolo[3,2-h]quinazoline-7-carboxamide
Canonical SMILESCSc1ncc2ccc3c(C(N)=O)c(C)n(C(C)C)c3c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P33981 TTK Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB