Molecule Details
InChIKeyPRIKHRTWFXDNDC-UHFFFAOYSA-N
Compound Name2-(3-methoxyphenyl)-N-(4-pyridin-4-ylthiophen-2-yl)acetamide
Canonical SMILESCOc1cccc(CC(=O)Nc2cc(-c3ccncc3)cs2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 8.0 Ki ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB
P17612 PRKACA Homo sapiens Human PF00069 6.2 Ki ChEMBL;BindingDB