Molecule Details
InChIKeyPREQLWGLUIHGJV-UHFFFAOYSA-N
Compound NameN-(6-chloro-7-fluoro-5-phenyl-1H-indazol-3-yl)butyramide
Canonical SMILESCCCC(=O)Nc1n[nH]c2c(F)c(Cl)c(-c3ccccc3)cc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.22
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget