Molecule Details
InChIKeyPQSAXJVMRVYGLM-UHFFFAOYSA-N
Compound Name4-[1-[3-[(3,3-Difluorocyclobutanecarbonyl)amino]phenyl]propylamino]quinazoline-8-carboxamide
Canonical SMILESCCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)C2CC(F)(F)C2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.7 IC50 ChEMBL;BindingDB