Molecule Details
InChIKeyPQOWYSIMYNJTLG-NEKODSHDSA-N
Compound Name(S)-2-[(S)-2-((S)-3-Carbamoyl-2-{(S)-3-methyl-2-[(S)-3-methyl-2-((R)-2-methyl-3-phenyl-propionylamino)-butyrylamino]-butyrylamino}-propionylamino)-3-carboxy-propionylamino]-4-methyl-pentanoic acid
Canonical SMILESCC(C)C[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](C)Cc1ccccc1)C(C)C)C(C)C)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23921 RRM1 Homo sapiens Human PF03477 PF02867 PF00317 6.1 IC50 ChEMBL;BindingDB
P31350 RRM2 Homo sapiens Human PF00268 6.1 IC50 ChEMBL
Q7LG56 RRM2B Homo sapiens Human PF00268 6.1 IC50 ChEMBL