Molecule Details
InChIKeyPPZARYOCIWUJNS-UHFFFAOYSA-N
Compound Name5-[3-(2-Methoxyphenyl)propyl]-2-phenylpyrazolo[4,3-d]pyrimidin-7-amine
Canonical SMILESCOc1ccccc1CCCc1nc(N)c2nn(-c3ccccc3)cc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 6.4 IC50 ChEMBL;BindingDB