Molecule Details
InChIKeyPPWZJWBTTSZJNT-UHFFFAOYSA-N
Compound NameN1-hydroxy-N4-(4-methyl-3-(4-(pyridin-3-yl)thiazol-2-ylamino)phenyl)terephthalamide
Canonical SMILESCc1ccc(NC(=O)c2ccc(C(=O)NO)cc2)cc1Nc1ncc(-c2cccnc2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.86
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.0 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.8 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.8 pIC50 TTD_MultiTarget