Molecule Details
InChIKeyPPNHBWGLEUAQKU-BHTNCQBCSA-N
Compound Name2-[2-(2-{2-[2-(2-Acetylamino-3-carboxy-propionylamino)-4-carboxy-butyrylamino]-3,3-diphenyl-propionylamino}-4-methoxycarbonyl-butyrylamino)-3-cyclohexyl-propionylamino]-4,4-difluoro-butyric acid
Canonical SMILESCC(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](CC(F)F)C(=O)O)C(c1ccccc1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C1KIQ2 Hepacivirus hominis Pathogen PF02907 7.5 Ki ChEMBL
D2K2A8 NS4A Hepacivirus hominis Pathogen PF01006 7.5 Ki ChEMBL
A3EZI9 NS3 Hepacivirus hominis Pathogen PF07652 PF22027 PF02907 7.4 Ki ChEMBL;BindingDB