Molecule Details
InChIKeyPPILDDFMLSKYDE-UHFFFAOYSA-N
Canonical SMILESC=CC(=O)N1CCC(Oc2n[nH]c3ncc(-c4cn(-c5c(F)ccc(NS(=O)(=O)c6ccccc6)c5F)nn4)cc23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYL2 MAP3K20 Homo sapiens Human PF07714 PF07647 8.0 IC50 ChEMBL
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 6.6 IC50 ChEMBL