Molecule Details
InChIKeyPPELJLBDXLMTEW-MRXNPFEDSA-N
Compound NameMmp-8 inhibitor i
Canonical SMILESCOc1ccc(S(=O)(=O)N2Cc3ccccc3C[C@@H]2C(=O)NO)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P22894 MMP8 Homo sapiens Human PF00045 PF00413 PF01471 8.4 IC50 ChEMBL;BindingDB
P08254 MMP3 Homo sapiens Human PF00045 PF00413 PF01471 7.7 IC50 ChEMBL
P18843 nadE Escherichia coli (strain K12) Pathogen PF02540 6.5 pIC50 TTD_MultiTarget