Molecule Details
InChIKeyPOSGRZQCKOTBHE-LLVKDONJSA-N
Compound Name4-[3-[(2R)-2-[(6-bromo-2-pyridinyl)oxy]propyl]-2-methylimidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine
Canonical SMILESCc1nc2ccc(-c3cc(N)nc(N)c3)nc2n1C[C@@H](C)Oc1cccc(Br)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB