Molecule Details
InChIKeyPOCXNIFHHUXWMU-UHFFFAOYSA-N
Compound NameN-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)nicotinamide
Canonical SMILESO=C(NCCN1CCCN(CC2COc3ccccc3O2)CC1)c1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB