Molecule Details
InChIKeyPNZJIQBIMCZAKU-UHFFFAOYSA-N
Compound Name2-[4-(Aminomethyl)piperidin-1-yl]-6-[2-(cyclohexylamino)-4-pyridinyl]pyridine-4-carboxamide
Canonical SMILESNCC1CCN(c2cc(C(N)=O)cc(-c3ccnc(NC4CCCCC4)c3)n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.89
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15139 PRKD1 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 7.3 IC50 ChEMBL;BindingDB
Q13563 PKD2 Homo sapiens Human PF18109 PF08016 PF20519 6.7 IC50 BindingDB
Q9BZL6 PRKD2 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 6.7 IC50 ChEMBL